Effectors: |
---|
1 | EFF0117 | Burton's tyrosine kinase-Homo sapiens-1 | Stimulation (indirect stimulation of p38 MAPK) | 15251227 | 9305846 | 16182515 |
2 | EFF0118 | Burton's tyrosine kinase-Homo sapiens-2 | Stimulation (indirect stimulation of p38 MAPK) | 15251227 | 9305846 | 16182515 |
3 | EFF0120 | Burton's tyrosine kinase-Homo sapiens-3 | Stimulation (indirect stimulation of p38 MAPK) | 15251227 | 9305846 | 16182515 |
4 | EFF0121 | Burton's tyrosine kinase-Homo sapiens-4 | Stimulation (indirect stimulation of p38 MAPK) | 15251227 | 9305846 | 16182515 |
5 | EFF0122 | Burton's tyrosine kinase-Homo sapiens-5 | Stimulation (indirect stimulation of p38 MAPK) | 15251227 | 9305846 | 16182515 |
6 | EFF0123 | Burton's tyrosine kinase-Homo sapiens-6 | Stimulation (indirect stimulation of p38 MAPK) | 15251227 | 9305846 | 16182515 |
7 | EFF0124 | Burton's tyrosine kinase-Homo sapiens-7 | Stimulation (indirect stimulation of p38 MAPK) | 15251227 | 9305846 | 16182515 |
8 | EFF0125 | Burton's tyrosine kinase-Homo sapiens-8 | Stimulation (indirect stimulation of p38 MAPK) | 15251227 | 9305846 | 16182515 |
9 | EFF0291 | Caveolin-1-Homo sapiens-1 | Gq Binds Caveolin to Concentrate in Caveolae | 16182515 | 11251080 |
10 | EFF0292 | Caveolin-1-Homo sapiens-2 | Gq Binds Caveolin to Concentrate in Caveolae | 16182515 | 11251080 |
11 | EFF0335 | EBP50/NHERF-1-Homo sapiens | Inhibits PLC-beta activation and blocks Gqa-induce Tph and CXCR4 receptor internalization | 16182515 |
12 | EFF0350 | GRK2-Homo sapiens | Inhibits PLC-beta activation and blocks Gqa-mediated GLUT4 translocation and glucose uptake in 3T3 adipocytes | 15251227 | 14654303 | 16182515 |
13 | EFF0359 | GRK3-Homo sapiens-1 | Stimulation | 15251227 | 14654303 | 16182515 |
14 | EFF0360 | GRK3-Homo sapiens-2 | Stimulation | 15251227 | 14654303 | 16182515 |
15 | EFF0397 | Kir 3.1(GIRK1)-Homo sapiens-1 | Inhibition | 12661754 |
16 | EFF0398 | Kir 3.1(GIRK1)-Homo sapiens-2 | Inhibition | 12661754 |
17 | EFF0410 | Kir 3.2(GIRK2)-Homo sapiens | Inhibition | 12661754 |
18 | EFF0420 | Kir 3.3(GIRK3)-Homo sapiens | Inhibition | 12661754 |
19 | EFF0425 | Kir 3.4(GIRK4)-Homo sapiens-1 | Inhibition | 12661754 |
20 | EFF0426 | Kir 3.4(GIRK4)-Homo sapiens-2 | Inhibition | 12661754 |
21 | EFF0434 | LARG RhoGEF-Homo sapiens-1 | Stimulation (indirect activation of Rho) | 15251227 | 12024019 |
22 | EFF0435 | LARG RhoGEF-Homo sapiens-2 | Stimulation (indirect activation of Rho) | 15251227 | 12024019 |
23 | EFF0442 | Lbc RhoGEF-Homo sapiens | No functional effects identified | 16182515 |
24 | EFF0443 | p115 RhoGEF-Homo sapiens | No data | 1525227 | 16182515 |
25 | EFF0444 | PDZ RhoGEF-Homo sapiens-1 | No data | 1525227 | 16182515 |
26 | EFF0445 | PDZ RhoGEF-Homo sapiens-2 | No data | 1525227 | 16182515 |
27 | EFF0517 | Phospholipase C beta-1-Homo sapiens-1 | Stimulation of PLC-beta catalytic activity | 15251227 | 16182515 | 11015615 |
28 | EFF0521 | Phospholipase C beta-1-Homo sapiens-2 | Stimulation of PLC-beta catalytic activity | 15251227 | 16182515 | 11015615 |
29 | EFF0522 | Phospholipase C beta-1-Homo sapiens-3 | Stimulation of PLC-beta catalytic activity | 15251227 | 16182515 | 11015615 |
30 | EFF0530 | Phospholipase C beta-2-Homo sapiens-1 | Stimulation of PLC-beta catalytic activity | 15251227 | 16182515 | 11015615 |
31 | EFF0531 | Phospholipase C beta-2-Homo sapiens-2 | Stimulation of PLC-beta catalytic activity | 15251227 | 16182515 | 11015615 |
32 | EFF0541 | Phospholipase C beta-3-Homo sapiens-1 | Stimulation of PLC-beta catalytic activity | 15251227 | 16182515 | 11015615 |
33 | EFF0542 | Phospholipase C beta-3-Homo sapiens-2 | Stimulation of PLC-beta catalytic activity | 15251227 | 16182515 | 11015615 |
34 | EFF0556 | Phospholipase C beta-4-Homo sapiens-1 | Stimulation of PLC-beta catalytic activity | 15251227 | 16182515 | 11015615 |
35 | EFF0558 | Phospholipase C beta-4-Homo sapiens-2 | Stimulation of PLC-beta catalytic activity | 15251227 | 16182515 | 11015615 |
36 | EFF0560 | Phospholipase C beta-4-Homo sapiens-3 | Stimulation of PLC-beta catalytic activity | 15251227 | 16182515 | 11015615 |
37 | EFF0572 | PI3K alpha-Homo sapiens | Inhibition of PI3K kinase activity in vitro | 16182515 |
38 | EFF0577 | PI3K beta-Homo sapiens-1 | Inhibition of PI3K kinase activity in vitro | 16182515 |
39 | EFF0578 | PI3K beta-Homo sapiens-2 | Inhibition of PI3K kinase activity in vitro | 16182515 |
40 | EFF0586 | PI3K gamma-Homo sapiens | Inhibition of PI3K kinase activity in vitro | 16182515 |
41 | EFF0595 | Protein kinase D-Homo sapiens | Stimulation | 10636921 |
42 | EFF0874 | Synembryn(Ric8a)-Homo sapiens | Stimulates Gqa activation and steady-state GTPase activity in vitro | 16182515 | 12509430 |
43 | EFF0877 | TRP repeat protein-1-Homo sapiens | G16a co-expression enhances TPR1 interaction with Ras | 16182515 | 12748287 |
44 | EFF1126 | Tubulin-Homo sapiens-1 | Potentiates receptor-induced PLC-beta activation | 16182515 |
45 | EFF1127 | Tubulin-Homo sapiens-10 | Potentiates receptor-induced PLC-beta activation | 16182515 |
46 | EFF1128 | Tubulin-Homo sapiens-11 | Potentiates receptor-induced PLC-beta activation | 16182515 |
47 | EFF1129 | Tubulin-Homo sapiens-12 | Potentiates receptor-induced PLC-beta activation | 16182515 |
48 | EFF1130 | Tubulin-Homo sapiens-13 | Potentiates receptor-induced PLC-beta activation | 16182515 |
49 | EFF1131 | Tubulin-Homo sapiens-14 | Potentiates receptor-induced PLC-beta activation | 16182515 |
50 | EFF1132 | Tubulin-Homo sapiens-15 | Potentiates receptor-induced PLC-beta activation | 16182515 |
51 | EFF1133 | Tubulin-Homo sapiens-16 | Potentiates receptor-induced PLC-beta activation | 16182515 |
52 | EFF1134 | Tubulin-Homo sapiens-17 | Potentiates receptor-induced PLC-beta activation | 16182515 |
53 | EFF1135 | Tubulin-Homo sapiens-18 | Potentiates receptor-induced PLC-beta activation | 16182515 |
54 | EFF1136 | Tubulin-Homo sapiens-19 | Potentiates receptor-induced PLC-beta activation | 16182515 |
55 | EFF1137 | Tubulin-Homo sapiens-2 | Potentiates receptor-induced PLC-beta activation | 16182515 |
56 | EFF1138 | Tubulin-Homo sapiens-20 | Potentiates receptor-induced PLC-beta activation | 16182515 |
57 | EFF1139 | Tubulin-Homo sapiens-21 | Potentiates receptor-induced PLC-beta activation | 16182515 |
58 | EFF1140 | Tubulin-Homo sapiens-22 | Potentiates receptor-induced PLC-beta activation | 16182515 |
59 | EFF1141 | Tubulin-Homo sapiens-23 | Potentiates receptor-induced PLC-beta activation | 16182515 |
60 | EFF1143 | Tubulin-Homo sapiens-25 | Potentiates receptor-induced PLC-beta activation | 16182515 |
61 | EFF1144 | Tubulin-Homo sapiens-26 | Potentiates receptor-induced PLC-beta activation | 16182515 |
62 | EFF1145 | Tubulin-Homo sapiens-27 | Potentiates receptor-induced PLC-beta activation | 16182515 |
63 | EFF1146 | Tubulin-Homo sapiens-28 | Potentiates receptor-induced PLC-beta activation | 16182515 |
64 | EFF1148 | Tubulin-Homo sapiens-3 | Potentiates receptor-induced PLC-beta activation | 16182515 |
65 | EFF1149 | Tubulin-Homo sapiens-30 | Potentiates receptor-induced PLC-beta activation | 16182515 |
66 | EFF1150 | Tubulin-Homo sapiens-31 | Potentiates receptor-induced PLC-beta activation | 16182515 |
67 | EFF1151 | Tubulin-Homo sapiens-32 | Potentiates receptor-induced PLC-beta activation | 16182515 |
68 | EFF1152 | Tubulin-Homo sapiens-33 | Potentiates receptor-induced PLC-beta activation | 16182515 |
69 | EFF1153 | Tubulin-Homo sapiens-34 | Potentiates receptor-induced PLC-beta activation | 16182515 |
70 | EFF1154 | Tubulin-Homo sapiens-35 | Potentiates receptor-induced PLC-beta activation | 16182515 |
71 | EFF1156 | Tubulin-Homo sapiens-37 | Potentiates receptor-induced PLC-beta activation | 16182515 |
72 | EFF1157 | Tubulin-Homo sapiens-38 | Potentiates receptor-induced PLC-beta activation | 16182515 |
73 | EFF1158 | Tubulin-Homo sapiens-39 | Potentiates receptor-induced PLC-beta activation | 16182515 |
74 | EFF1159 | Tubulin-Homo sapiens-4 | Potentiates receptor-induced PLC-beta activation | 16182515 |
75 | EFF1160 | Tubulin-Homo sapiens-40 | Potentiates receptor-induced PLC-beta activation | 16182515 |
76 | EFF1162 | Tubulin-Homo sapiens-42 | Potentiates receptor-induced PLC-beta activation | 16182515 |
77 | EFF1163 | Tubulin-Homo sapiens-43 | Potentiates receptor-induced PLC-beta activation | 16182515 |
78 | EFF1164 | Tubulin-Homo sapiens-44 | Potentiates receptor-induced PLC-beta activation | 16182515 |
79 | EFF1165 | Tubulin-Homo sapiens-45 | Potentiates receptor-induced PLC-beta activation | 16182515 |
80 | EFF1166 | Tubulin-Homo sapiens-46 | Potentiates receptor-induced PLC-beta activation | 16182515 |
81 | EFF1167 | Tubulin-Homo sapiens-47 | Potentiates receptor-induced PLC-beta activation | 16182515 |
82 | EFF1168 | Tubulin-Homo sapiens-48 | Potentiates receptor-induced PLC-beta activation | 16182515 |
83 | EFF1169 | Tubulin-Homo sapiens-49 | Potentiates receptor-induced PLC-beta activation | 16182515 |
84 | EFF1170 | Tubulin-Homo sapiens-5 | Potentiates receptor-induced PLC-beta activation | 16182515 |
85 | EFF1171 | Tubulin-Homo sapiens-50 | Potentiates receptor-induced PLC-beta activation | 16182515 |
86 | EFF1173 | Tubulin-Homo sapiens-52 | Potentiates receptor-induced PLC-beta activation | 16182515 |
87 | EFF1174 | Tubulin-Homo sapiens-51 | Potentiates receptor-induced PLC-beta activation | 16182515 |
88 | EFF1175 | Tubulin-Homo sapiens-41 | Potentiates receptor-induced PLC-beta activation | 16182515 |
89 | EFF1176 | Tubulin-Homo sapiens-36 | Potentiates receptor-induced PLC-beta activation | 16182515 |
90 | EFF1177 | Tubulin-Homo sapiens-29 | Potentiates receptor-induced PLC-beta activation | 16182515 |
91 | EFF1178 | Tubulin-Homo sapiens-24 | Potentiates receptor-induced PLC-beta activation | 16182515 |
92 | EFF1179 | Tubulin-Homo sapiens-6 | Potentiates receptor-induced PLC-beta activation | 16182515 |
93 | EFF1180 | Tubulin-Homo sapiens-7 | Potentiates receptor-induced PLC-beta activation | 16182515 |
94 | EFF1181 | Tubulin-Homo sapiens-8 | Potentiates receptor-induced PLC-beta activation | 16182515 |
95 | EFF1182 | Tubulin-Homo sapiens-9 | Potentiates receptor-induced PLC-beta activation | 16182515 |